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RSS Feeds[ASAP] Determination of Ligand Binding Epitope Structures Using Polarization Transfer from Hyperpolarized Ligands (Journal of Medicinal Chemistry)

 
 

21 february 2019 01:03:32

 
[ASAP] Determination of Ligand Binding Epitope Structures Using Polarization Transfer from Hyperpolarized Ligands (Journal of Medicinal Chemistry)
 


Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.8b01711


 
48 viewsCategory: Chemistry, Medicine
 
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[ASAP] Exploiting the Tolerant Region I of the Non-Nucleoside Reverse Transcriptase Inhibitor (NNRTI) Binding Pocket: Discovery of Potent Diarylpyrimidine-Typed HIV-1 NNRTIs against Wild-Type and E138K Mutant Virus with Significantly Improved Water Solubility and Favorable Safety Profiles (Journal of Medicinal Chemistry)
 
 
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