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RSS Feeds[ASAP] Fluorination of Photoswitchable Muscarinic Agonists Tunes Receptor Pharmacology and Photochromic Properties (Journal of Medicinal Chemistry)

 
 

19 march 2019 18:00:02

 
[ASAP] Fluorination of Photoswitchable Muscarinic Agonists Tunes Receptor Pharmacology and Photochromic Properties (Journal of Medicinal Chemistry)
 


Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.8b01822


 
54 viewsCategory: Chemistry, Medicine
 
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[ASAP] Optimization of P2Y12 Antagonist Ethyl 6-(4-((Benzylsulfonyl)carbamoyl)piperidin-1-yl)-5-cyano-2-methylnicotinate (AZD1283) Led to the Discovery of an Oral Antiplatelet Agent with Improved Druglike Properties (Journal of Medicinal Chemistry)
 
 
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