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RSS Feeds[ASAP] Multistage Screening Reveals 3-Substituted Indolin-2-one Derivatives as Novel and Isoform-Selective c-Jun N-terminal Kinase 3 (JNK3) Inhibitors: Implications to Drug Discovery for Potential Treatment of Neurodegenerative Diseases (Journal of Medicinal Chemistry)

 
 

16 july 2019 03:01:21

 
[ASAP] Multistage Screening Reveals 3-Substituted Indolin-2-one Derivatives as Novel and Isoform-Selective c-Jun N-terminal Kinase 3 (JNK3) Inhibitors: Implications to Drug Discovery for Potential Treatment of Neurodegenerative Diseases (Journal of Medicinal Chemistry)
 


Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.9b00537


 
179 viewsCategory: Chemistry, Medicine
 
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[ASAP] Discovery of a Thiadiazole-Pyridazine-Based Allosteric Glutaminase 1 Inhibitor Series That Demonstrates Oral Bioavailability and Activity in Tumor Xenograft Models (Journal of Medicinal Chemistry)
 
 
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