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RSS Feeds[ASAP] Discovery of a Thiadiazole-Pyridazine-Based Allosteric Glutaminase 1 Inhibitor Series That Demonstrates Oral Bioavailability and Activity in Tumor Xenograft Models (Journal of Medicinal Chemistry)

 
 

17 july 2019 05:00:20

 
[ASAP] Discovery of a Thiadiazole-Pyridazine-Based Allosteric Glutaminase 1 Inhibitor Series That Demonstrates Oral Bioavailability and Activity in Tumor Xenograft Models (Journal of Medicinal Chemistry)
 


Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.9b00260


 
202 viewsCategory: Chemistry, Medicine
 
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[ASAP] Novel Human Aminopeptidase N Inhibitors: Discovery and Optimization of Subsite Binding Interactions (Journal of Medicinal Chemistry)
 
 
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